Enzymatic activation of a matrix metalloproteinase inhibitor.
نویسندگان
چکیده
Matrix metalloproteinase inhibitors (MMPi) possessing a glucose protecting group on the zinc-binding group (ZBG) show a dramatic increase in inhibitory activity upon cleavage by beta-glucosidase.
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ورودعنوان ژورنال:
- Chemical communications
دوره 46 8 شماره
صفحات -
تاریخ انتشار 2010